Immense opportunities of customization
to meet each project’s specific needs
○ Targets: GPCRs, kinases, NHR, transporters, ion channels, protease
○ Readouts: ELISA, reporter, binding, internalization, proliferation,
chemotaxis, 2nd messenger, flow cytometry, chemiluminescence,
TR-FRET, absorbance, and radioisotope
○ Modalities: agonist (full, partial, inverse), antagonist (full, partial), allosteric modulators (PAM, NAM)